bilastine

bilastine

Clinical data
Trade names	Blexten, others
Pregnancy category	AU: B3
Routes of administration	By mouth
Drug class	Antihistamine
ATC code	R06AX29 (WHO) S01GX13 (WHO)
Legal status
Legal status	AU: S2 (Pharmacy medicine) CA: ℞-only NZ: S2 (Pharmacy Only)
Pharmacokinetic data
Bioavailability	61%
Protein binding	84-90% binding to plasma proteins
Metabolism	Not significantly metabolised
Onset of action	1 hour (Allertine)
Elimination half-life	14.5 hours
Duration of action	24 hours (Allertine)
Excretion	95% in urine and faeces
Identifiers
IUPAC name 2-[4-(2-{4-[1-(2-Ethoxyethyl)-1H-benzimidazol-2-yl]-1-piperidinyl}ethyl)phenyl]-2-methylpropanoic acid
CAS Number	202189-78-4 Y
PubChem CID	185460
DrugBank	DB11591
ChemSpider	161234 Y
UNII	PA1123N395
KEGG	D09570
ChEMBL	ChEMBL1742423 Y
Chemical and physical data
Formula	C28H37N3O3
Molar mass	463.622 g·mol−1
3D model (JSmol)	Interactive image
SMILES O=C(O)C(c1ccc(cc1)CCN4CCC(c2nc3ccccc3n2CCOCC)CC4)(C)C
InChI InChI=1S/C28H37N3O3/c1-4-34-20-19-31-25-8-6-5-7-24(25)29-26(31)22-14-17-30(18-15-22)16-13-21-9-11-23(12-10-21)28(2,3)27(32)33/h5-12,22H,4,13-20H2,1-3H3,(H,32,33) Y Key:ACCMWZWAEFYUGZ-UHFFFAOYSA-N Y
NY (what is this?)  (verify)

Angol

Főnév

bilastine (tsz. bilastines)

1. (gyógyszertan) bilasztin

További információk

• bilastine - Szótár.net (en-hu)
• bilastine - Sztaki (en-hu)
• bilastine - Merriam–Webster
• bilastine - Cambridge
• bilastine - WordNet
• bilastine - Яндекс (en-ru)
• bilastine - Google (en-hu)
• bilastine - Wikidata
• bilastine - Wikipédia (angol)