gepirone

gepirone

Clinical data
Trade names	Exxua
Other names	BMY-13805; MJ-13805; ORG-13011
Routes of administration	By mouth
ATC code	N06AX19 (WHO)
Legal status
Legal status	US: ℞-only
Pharmacokinetic data
Bioavailability	14–17%
Protein binding	72%
Metabolism	CYP3A4
Metabolites	3'-OH-gepirone; 1-(2-Pyrimidinyl)piperazine
Elimination half-life	IRTooltip Instant release: 2–3 hours ERTooltip Modified-release dosage: 5 hours
Excretion	Urine: 81%
Identifiers
IUPAC name 4,4-Dimethyl-1-[4-(4-pyrimidin-2-ylpiperazin-1-yl)butyl]piperidine-2,6-dione
CAS Number	83928-76-1 Y 83928-66-9
PubChem CID	55191
DrugBank	DB12184 DBSALT002148
ChemSpider	49836 Y 49835
UNII	JW5Y7B8Z18 80C9L8EP6V
KEGG	D04314
ChEBI	CHEBI:135990
ChEMBL	ChEMBL284092 Y ChEMBL1204187
Chemical and physical data
Formula	C19H29N5O2
Molar mass	359.474 g·mol−1
3D model (JSmol)	Interactive image
SMILES O=C1N(C(=O)CC(C)(C)C1)CCCCN3CCN(c2ncccn2)CC3
InChI InChI=1S/C19H29N5O2/c1-19(2)14-16(25)24(17(26)15-19)9-4-3-8-22-10-12-23(13-11-22)18-20-6-5-7-21-18/h5-7H,3-4,8-15H2,1-2H3 Y Key:QOIGKGMMAGJZNZ-UHFFFAOYSA-N Y
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Angol

Főnév

gepirone (tsz. gepirones)

1. (gyógyszertan) gepiron

További információk

• gepirone - Szótár.net (en-hu)
• gepirone - Sztaki (en-hu)
• gepirone - Merriam–Webster
• gepirone - Cambridge
• gepirone - WordNet
• gepirone - Яндекс (en-ru)
• gepirone - Google (en-hu)
• gepirone - Wikidata
• gepirone - Wikipédia (angol)